Medicinal Chemistry

(Jacob Rumans) #1

P. M. Laduron (1982). Towards a unitary concept of opiate receptor. Trends Pharmacol. Sci. 3:
351–352.
K. E. Light (1984). Analyzing non-linear Scatchard plots. Science 223: 76–77.


Receptor Binding Terms


E. J. Ariëns (1983). Intrinsic activity: partial agonists and partial antagonists. J. Cardiovasc.
Pharmacol. 5: S8–SI5.
F. J. Barrantes (1979). Endogenous chemical receptors: some physical aspects. Annu. Rev.
Biophys. Bioeng. 8 : 287–321.
J. M. Boeynaems, J. E. Dumont (Eds.) (1980). Outlines of Receptor Theory. New York:
Elsevier/North Holland.
J. P. Changeux (1995). The acetylcholine receptor: A model for allosteric membrane proteins.
Biochem. Soc. Trans. 23: 195.
D. Colquhoun (1973). The relation between classical and cooperative models for drug action. In:
H. P. Rang (Ed.).Drug Receptors. Baltimore: University Park Press, pp. 149–182.
A. De Lean, P. J. Munson, D. Rodbard (1979). Multivalent ligand binding to multisubsite recep-
tors: application to hormone–receptor interactions. Mol. Pharmacol. 15: 60–70.
A. De Lean, D. Rodbard (1979). Kinetics of cooperative binding. In: R. D. O’Brien (Ed.). The
Receptors. New York: Plenum Press, pp. 143–192.
J. DiMaio, F. R. Ahmed, P. Shiller, B. Belleau (1979). Stereo-electronic control and decontrol of
the opiate receptor. In: F. Gualtieri, M. Gianella, and C. Melchiorre (Eds.). Recent Advances
in Receptor Chemistry. New York: Elsevier/North Holland, pp. 221–234.
M. D. Hollenberg, P. Cuatrecasas (1979). Distinction of receptor from non-receptor interaction in
binding studies. In: R. D. O’Brien (Ed.). The Receptors. New York: Plenum Press, pp. 193–214.
P. M. Laduron (1984). Criteria for receptor sites in binding studies. Biochem. Pharmacol. 33 :
833–839.
D. E. Macfarlane (1984). On the enzymatic nature of receptors. Trends Pharmacol. Sci. 5 : 11–15.
H. G. Mautner (1980). Receptor theories and dose–response relationships. In: M. E. Wolff (Ed.).
The BasisofMedicinal Chemistry,4th ed., vol. 1. New York: Wiley-Interscience, pp. 271–284.
M. Poo (1985). Mobility and localization of proteins in excitable membranes. Annu. Rev.
Neurosci. 8: 369–406.
D. Rodbard (1980). Agonist versus antagonist. Trends Pharmacol. Sci. 1: 222–225.
K. Starke (1981). Presynaptic receptors. Annu. Rev. Pharmacol. Toxicol. 21: 7–30.
R. P. Stephenson (1956). A modification of receptor theory. Br. J. Pharmacol. 11 : 379–393.
D. J. Triggle, C. R. Triggle (1976). Chemical Pharmacologyofthe Synapse. New York: Academic
Press, chapter 2.


Receptor Metabolism


J. L. Carpentier, P. Gorden, A. Roberts, L. Orci (1986). Internalization of polypeptide hormones
and receptor cycling. Experientia 42: 734–744.
R. B. Dickson (1985). Endocytosis of polypeptides and their receptors. Trends Pharmacol. Sci.
6 : 164–167.
I. A. Hanover, R. B. Dickson (1985). The possible link between receptor phosphorylation and
internalization.Trends Pharmacol. Sci. 6: 457–459.
M. D. Hollenberg (1985). Receptor regulation, Parts 1 and 2. Trends Pharmacol. Sci. 6: 242–245;
299–302.
J. A. Koenig, J. Edwardson (1997). Endocytosis and recycling of G protein receptors. Trends
Pharmacol Sci. 18: 276.


104 MEDICINAL CHEMISTRY

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