Medicinal Chemistry

(Jacob Rumans) #1

Estrogen/progestin replacement
therapy


ESTROGENS,ORAL
conjugated estrogens
estradiol-17β
estropipate
ethinyl estradiol


ESTROGENS,PARENTERAL
estradiol valerate


ESTROGENS,TRANSDERMAL
estradiol-17β


ESTROGENS,VAGINAL PREPARATIONS
conjugated estrogens
estradiol
estradiol-17βhemihydrate
estrone


PROGESTOGENS
medrogestone
medroxypogesterone acetate
megestrol acetate
norethindrone


ESTROGEN/PROGESTOGEN
COMBINATIONS,ORAL
conjugated estrogens/
medroxyprogesterone
ethinyl estradiol/norethindrone acetate
mestranol/norethindrone


ESTROGEN/PROGESTOGEN COMBINATIONS,
TRANSDERMAL
estradiol-17β/norethindrone


Hypercalcemia and Paget’s disease


Bone metabolism regulators


ANTIPARATHYROID HORMONES
calcitonin salmon


BISPHOSPHONATES
alendronate sodium
clodronate disodium
etidronate disodium
pamidronate disodium
risedronate sodium
zoledronic acid


PHOSPHATE PREPARATIONS

sodium acid phosphate

Hypothalamic and pituitary
hormones
(see also Cancer, hormones;
Endometriosis; Hormonal therapy;
Thyroid disorders)
Anterior pituitary hormones
ADRENOCORTICOTROPHIC HORMONES
(ACTH)
cosyntropin
cosyntropin/zinc hydroxide

GROWTH HORMONES
somatrem
somatropin

Hypothalamic hormones
GONADOTROPIN-RELEASING HORMONE
(GNRH)ANALOGS
buserelin acetate
goserelin acetate
leuprolide acetate
nafarelin acetate

SOMATOSTATIN AND ANALOGS
octreotide acetate
somatostatin

Posterior pituitary hormones
ANTIDIURETIC HORMONE ANALOGS
desmopressin acetate
vasopressin
OXYTOCICS
oxytocin

Infertility
GONADOTROPINS
follitropin alpha (rDNA origin)
follitropin beta (rec FSH)
gonadotropin (human) chorionic
menotropins
GONADOTROPIN-RELEASING HORMONE
ANTAGONISTS
ganirelix acetate

606 MEDICINAL CHEMISTRY

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