Medicinal Chemistry

(Jacob Rumans) #1

Bleeding therapy


Antifibrinolytics


AMINO ACIDS
aminocaproic acid
tranexamic acid


PROTEINASE INHIBITORS
aprotinin


VITAMINKANALOGUES
phytonadione


Hemostatics


BLOOD COAGULATION FACTORS
antihemophilic factor (recombinant)
eptacog alfa (activated)
factor IX contentrate (human)
factor IX (recombinant)
moroctocog alfa


LOCAL HEMOSTATICS
thrombin (bovine)
gelatin, absorbable


VARIOUS HEMOSTATICS
desmopressin acetate


Mineral replacement


Iron replacement therapy


IRON BIVALENT,ORAL PREPARATIONS
ferrous fumarate
ferrous gluconate
ferrous sulfate


IRON TRIVALENT,PARENTERAL PREPARATIONS
iron sorbitol citric acid complex


Platelet antiaggregation therapy


ADENOSINE DIPHOSPHATE INHIBITORS
clopidogrel bisulfate
dipyridamole
sulfinpyrazone


GLYCOPROTEIN(GPLLB/LLLA)
RECEPTOR INHIBITORS
abciximab
eptifibatide
tirofiban hydrochloride


FIBRINOGEN-PLATELET BINDING INHIBITORS

ticlipidine hydrochloride
THROMBOXANE-A 2 INHIBITORS
acetylsalicylic acid (ASA)

Thrombolytic therapy
Plasminogen activators
NATURALENZYMES
urokinase
PROTEINS,DERIVED FROM BACTERIA
reteplase
streptokinase
PROTEINS,RECOMBINANT
DNA ORIGIN
alteplase
anistreplase
tenecteplase
VARIOUS ANTITHROMBOTIC AGENTS
anagrelide hydrochloride
fondaparins sodium

IMMUNOLOGY

Corticosteroid therapy, systemic
GLUCOCORTICOIDS
betamethasone acetate
betamethasone sodium phosphate
cortisone acetate
dexamethasone
dexamethasone sodium
phosphate
hydrocortisone
hydrocortisone sodium succinate
methylprednisolone acetate
methylprednisolone sodium
succinate
prednisolone sodium phosphate
prednisone
triamcinolone
triamcinolone acetonide
triamcinolone diacetate
MINERALOCORTICOIDS
fludrocortisone acetate

DRUGS ARRANGED BY PHARMACOLOGIC ACTIVITY 611
Free download pdf