Organic Chemistry of Drug Synthesis. Volume 7

(Brent) #1

Antibacterial(Continued)
Sitafloxacin, 174
Antidepressant
Citalopram, 140
Elzasonan, 136
Flibanserin, 158
Igmesine, 64
Lubazodone, 70
Reboxetine, 61
Vofopitant, 110
Antidiabetic
Ertiprotafib, 219
Muraglitazar, 47
Nateglinide, 15
Netoglitazone, 103
Ragaglitazar, 220
Repaglinide, 15
Rivoglitazone, 157
Sitagliptan, 206
Vidagliptin, 84
Antiemetic
Aprepitant, 105
Ezlopitant, 62
Maropitant, 62
Antiepileptic
Rufinamide, 108
Antiestrogen
Acolbifene, 163
Arzoxyfene, 155
Bazedoxifene, 145
Fulvestrant, 32
Lasofoxifene, 77
Ospemifene, 65
Antifungal
Omoconazole, 94
Posaconazole, 105
Voriconazole, 103
Antihpertensive
Atrasentan, 87
Gemopatrilat, 19
Clevipidine, 117
Edonentan, 56
Nepicastat, 97
Olmesartan, 111
Antiinflammatory
Darbufelone, 99
Ecopladib, 147
Pelitinib, 167


Varespladib, 144
Antiinflammatory COX-2
Cimicoxib, 96
Etoricoxib, 117
Parecoxib, 92
Tilmacoxib, 91
Valdecoxib, 92
Antiparasitic
Nitazoxinide, 101
Antiprogestin
Asoprinosil, 32
Antipsychotic
Asenapine, 228
Bifeprunox, 159
Ecopipam, 228
Paliperidone, 209
Sonepiprazole, 166
Antitumor
Alitretoin, 30
Alvocidib, 165
Apaziquone, 154
Bexarotene, 76
Bortezomib, 133
Camptogen, 230
Canertinib, 180
Canfosfamide, 13
Clofarabine, 200
Cloretazine, 14
Doramapimod, 74
Emitefur, 127
Enzastaurin, 89
Erlotinib, 179
Exatecan, 232
Forodesine, 192
Gefitinib, 181
Irofulven, 38
Istradefylline, 202
Lapatinib, 182
Monasterol, 128
Mubritinib, 108
Nelarabine, 200
Pelitrexol, 212
Pemetrexed, 193
Pralatrexate, 211
Prinomastat, 54
Semaxanib, 149
Sunitinib, 150
Talabostat, 84

242 CROSS INDEX OF BIOLOGICAL ACTIVITY

Free download pdf