Exercise for Cardiovascular Disease Prevention and Treatment From Molecular to Clinical, Part 1

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7 Moderate Exercise Training (MET) and Stabilization


of Nrf2-Antioxidant Signaling in the Myocardium


Given the role of Nrf2 during short sub-maximal (acute) and maximal endurance


stress in aging animals, a moderate exercise training (MET) for a longer duration


(6 weeks) seems to significantly augment nuclear Nrf2 level in both the young and


aging heart. Subsequent to MET-induced Nrf2 stabilization, an increase in the tran-


script and protein levels of major Nrf2-targets (i.e. glutathione reductase, hemoxy-


genase- 1, glucose 6-phosphate dehydrogenase and glutamyl cysteine ligase) was


also demonstrated [ 75 ]. Prior studies have established that a short- and long-term


MET promoted myocardial perfusion and functional capacity in animals and


humans with ischemic heart disease, and heart failure [ 152 , 156 , 159 – 166 ]. Notably,


MET has been beneficial in preventing age-related cardiovascular diseases [ 15 ,


167 ]. We along with others have shown that, although there was an MET-induced


protection seen in aged animals the magnitude of benefits was not as strong as that


noted in the younger group [ 75 , 168 ]. However, the precise mechanisms are still


elusive. Based on our previous study, it can be agreed upon that moderate exercise


training in aging animals can escalate Nrf2 signaling and restore redox homeostasis


[ 75 ], but the inherently high oxidative burden that exists during aging could require


a much stronger Nrf2 activation and its associated antioxidant signaling than that is


currently offered by MET. In other words, optimal benefits of MET could depend


on the optimization of redox and this could be one of the crucial points where the


young and old diverge with respect to MET’s effect. Further, an interesting finding


has demonstrated that when animals were subjected to swimming in warm water at


30–32  °C with a duration of 60  min (5  days/week) for 10  weeks that represents


MET, showed neovascularization along with improved structure and function of the


cardiovascular system [ 169 – 171 ]. Although MET can enhance Nrf2 signaling in the


aging model, how far MET can be effective in improving the proangiogenic process


in aging is unclear currently. Since, it has been reported that Nrf2 can activate


HIF-1α/VEGF pathway [ 172 , 173 ], investigating the molecular cross-talk between


Nrf2 with angiogenesis in response to MET in young and aged hearts could also be


worthwhile to narrow the gap in our understanding along these lines. Nevertheless,


moderate exercise training is still the most preferred and applied training modality


for improving cardiac fitness. However, new training modes and/or strategies are in


need for the aged segment. With the current understanding, we suppose an in-depth


animal study involving a combination of MET along with a titrated nutraceutical or


dietary mode of Nrf2 activation through Protandim or Broccoli, that contains sul-


foraphane (an activator of Nrf2) respectively will be an ideal starting point. And,


hopefully, more studies in this line of thought can provide impetus to explore an


effective strategy to improve the cardiac fitness in the elderly.


M. Narasimhan and N.-S. Rajasekaran
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