AMPK Methods and Protocols

(Rick Simeone) #1

  1. The time and temperature for an IP can vary a lot depending on
    antibody affinity, considerations for protein complex stability,
    and workflow. Low temperature (4C) lengthens the IP pro-
    cess but maintains a higher stability for protease and phospha-
    tase inhibitors as well as for protein interactions. Doing
    consecutive IPs and measuring enzyme activity on each of the
    IPs would challenge the number of hours in a working day if
    the time for each IP was set to only a couple of hours. Our
    experience is that the AMPK heterotrimeric complexes are very
    stable and can endure at least three consecutive overnight IP
    incubations at 4C. We have assayed theα1-,α2-, andγ3-
    associated activities after 4 h and one, two, and three overnight
    incubations with similar results.

  2. The total volume of each of the firstγ3 IPs is 200μl of which
    10 μl is packed agarose beads and 190μl is supernatant. By only
    transferring 170μl to the next IP, protein is lost, but there
    must be a safety margin to avoid transferring agarose with
    bound AMPK to the next IP. The second IP (α2) will thus be
    on (250μg/190μl) 170μl¼ 224 μg total protein. The total
    volume of theα2 IP will be 200μl (20μl of Protein G agarose,
    10 μl of antibody, and 170μl of supernatant from theγ3 IP)
    like the first IP of which 190μl is supernatant. Transferring
    170 μl of supernatant from the secondα2 IP to the thirdα1IP
    will give this IP (224μg/190μl)
    170μl¼ 200 μg total
    protein. These amounts of total protein precipitated on (input)
    will be used in the calculations of the specific AMPK activities
    that are given as pmol ATP incorporated into the AMARA
    peptide per minute of time for the kinase reaction per mg lysate
    precipitated on (pmol/min/mg).

  3. When transferring the supernatant from one IP to the next,
    place the first PCR-plate on the table and use plenty of light.
    Place a mirror on one side of the PCR-plate, so you can see
    both the first pipette tip of the eight-channel pipette on the
    side facing you and the eighth tip facing the mirror. This way
    you will be sure that none of the eight pipette tips reach the
    agarose at the bottom of the wells. After the transfer of all
    supernatants, put the PCR-plate back on ice.

  4. The stock solutions for preparing the kinase reaction buffer are
    stored at 20 C unless otherwise indicated. We use the fol-
    lowing stock concentrations: 5 mM DTT, 2 mM AMP,
    1.5 mM AMARA peptide, 150 mM MgCl 2 (stored at 4C),
    10 mM ATP, and^33 P-ATP (10μCi/μl) (stored at 4C). In
    order to make up kinase reaction buffer for one sample (30μl),
    mix 8.3μl water, 5μl DTT, 3μl AMP, 2μl AMARA peptide,
    1 μl MgCl 2 , 0.6μl ATP, 0.1μl^33 P-ATP (on calibration date),
    and 10μl3Assay buffer (120 mM HEPES and 240 mM
    NaCl). The amount of water and^33 P-ATP depends on the


226 Jesper B. Birk and Jørgen F. P. Wojtaszewski

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