Fundamentals of Medicinal Chemistry

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particular drug, it is essential that the equipment used is cleaned and tested for

adulterants before use. Many pharmaceutical manufacturers estimated that

production line equipment is only used to produce the product for about 10%

of its time. For most of the remaining time it is being stripped down, cleaned and

reassembled.

The quality control of drugs and medicines during and after production is

essential for their safe use. It was only achieved when accurate analytical

methods were developed in the mid-19th century. This led to the publication

of national pharmacopoeias and other documents that specified the extent and

the nature of the identification tests and quantitative assessments required to

ensure that the product reaching the public is fit for its purpose. These docu-

ments now cover the production, storage and application of pharmaceutical

products. They are the subject of constant review but unfortunately this does

not completely prevent the occurrence of product related problems. However,

the continual updating of these documents does reduce the possibility of similar

problems occurring in other products. It is gratifying to note that since the

thalidomide disaster very few drugs have been removed from the market on

safety grounds. The development of reliable analytical methods for the trials,

production quality control and identification, limit and assay procedures for

inclusion into the relevant pharmacopoeias is normally carried out in parallel

to the critical path development stages. These analytical methods must be

described in detail in the product licence application.

11.7 Patent protection


The high cost of drug development and production makes it essential for a

company to maximize its returns from a new drug. This can only be achieved by

preventing unrestricted copying of a new product by rivals. Patents are used to

prevent rival companies manufacturing and marketing a product without the

permission of the originator of the product. However, many companies do

market other manufacturers’ products under licence from the original patentor.

Patents have been used, in one form or another, as a means of industrial

protection from the early 14th century to the present day. Originally, they were

intended to encourage the development of new industries and products by

granting the developer or producer the monopoly to either use specific industrial

equipment or produce specific goods for a limited period. This monopoly,

enforced by the appropriate government office, enabled an innovator to obtain

a just reward for his efforts. In most countries the awarding of a patent prevents

236 DRUG DEVELOPMENT AND PRODUCTION

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