Fundamentals of Medicinal Chemistry

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third parties from manufacturing and selling the product without the consent of

the innovator. However, patents do encourage and protect the development of

new ideas by the publication of new knowledge.

Originally each country issued its own patent laws, but by the mid-18th

century it was recognized that patent rights should extend beyond national

boundaries. The first international agreement was theParis Convention of

1883. This has been revised on numerous occasions, the current treaties in

operation being the Europeans Union’s European Patent Convention (EPC)

of 1978 and the Patent Cooperation Treaty (PCT) signed in Washington in

1970. The former is only open to European countries and administered by the

European Patents Office (EPO). The latter is open to all countries of the world

and is administered through the national patent offices of the country subscrib-

ing to the treaty.

The protection offered by a patent is of paramount importance to a company

at the research, development and production stages of drug production. It is

essential that a patent is filed as soon as new compounds have been made and

shown to have interesting properties. Otherwise, a rival company working in the

same field might pre-empt the patent, which means that a large amount of

expensive research work would be unproductive in respect to company profits.

In this respect, it is particularly important that the patent covers the relevant

field and does not give a rival manufacturer an exploitable loophole.

The time required for the development of a drug from discovery to produc-

tion can take at least 7–15 years. In many countries, patents normally run for 20

years from the date of application. Consequently, the time available for a

manufacturer to recoup the cost of development and show a profit is rather

limited, which accounts for the high cost of some new drugs. Furthermore, it

also means that some compounds are never developed because the patent

protected production time available to recoup the cost of development is too

short.

11.8 Regulation


The release of a new drug onto the market must be approved by the regulating

authority for that country. For example, in Britain this is the Medicines Control

Agency (MCA), in the European Union it is the European Medicines Evalu-

ation Agency (EMEA) and in the USA the US Food and Drugs Administration

(FDA). These bodies, which are essentially consumer protection agencies, issue

a so calledproduct licenceormarketing authority (MA)when they are satisfied

REGULATION 237

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