Medicinal Chemistry

Pain Nonsteroidal anti-inflammatory drugs (NSAIDs) ACETIC ACID DERIVATIVES(INCLUDING INDOLE DERIVATIVES) diclofenac potassium di ...

Ethylene glycol antidote ALCHOHOL DEHYDROGENASE INHIBITOR fomepizol HEPARIN ANTAGONISTS protamine sulfate Nonspecific therapy fo ...

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Index 629 Aβpeptide, 513, 515, 516 ab initio calculations, 46 abacavir, 555 abortion, threatened spontaneous, 326 absolute confi ...

alkylating agents, 446 allopurinol, 471 allosteric inhibition, 76, 484 allosteric site, 484 N-allyl-norcodeine, 358 Alzheimer’s ...

aromatic electrophilic substitution, 128 aromatic nucleophilic substitution, 128 arrhythmia, heart, 379, 420–421 arsenic poisoni ...

breast cancer, estrogen dependent, 325 bremazocine, 357 bretylium, 227 bromide therapy, 118 bromination of alkenes, 171 bromocri ...

Charles II, death, 109 cheilosis, 505 chelates, 594 cheminformatics, 61–63, 127 chemogenomics, 127 chemokines, 398–401 chemotact ...

cranial nerves, 199 cresol, 571 cretinism, 361 Creutzfeldt-Jakob disease, 100, 514, 515, 546 CRF, 288, 289, 332, 345–346 Crick, ...

dimaprit, 264 dimenhydrinate, 266 dimercaprol, 595 dimercaptopropane, 595 dipeptide, 338 diphenhydramine, 14, 266 diplopia, 512 ...

ergot alkaloids, 242, 349 ergotamine, 256 ERICE, 503 ERT, 537 erythema, 525 erythromycin, 18, 576 eserine, 488 essential oils, 4 ...

G-protein receptors, 92–96, 224, 284, 290 GABA, 270–273, 422, 432 GABA receptors, 271, 272 gabaculine, 272 gabapentin, 18, 279 G ...

Helicobacter pylori, 268 Hell-Volhard-Zellinski reaction, 172 helminths, 585 hemoglobin, 479 heparin, 16, 512, 528 heparins, low ...

inhibin, 316 inhibitory factors, 340 innate immunity, 390 inorganic substances as drugs and targets, 532–537 inosiplex, 397, 398 ...

Lineweaver-Burke, plot, 83 lipid peroxidation, 411 lipids, 471–474 as drugs and targets, 519 Lipinski’s rule, 10 lipoproteins, 3 ...

metals, 480–481 main group, 480 transition, 480 metastasis, 457, 461 metazocine, 357 metformin, 367, 368 methacholine, 210 metha ...

naphazoline, 229 naproxen, 525 natriptam, 260 natriuresis, 376 natriuretic factor, 311, 376–378 NE, 498 necrosis, 500, 501 nelfi ...

oligopeptide libraries, 123 oligosaccharide, 475 omeprazole, 268, 494 oncogenes, 95 Ondetti, 373 one target-multiple disease app ...

pH, tissue fluids, 13 phagocytosis, 390 pharmaceutical phase, 10–15 pharmacodynamic phase, 10, 17–19, 134–139 pharmacogenomics, ...

progestogens, 326 proglucagon, 371 progoitrin, 362 prohormones, 339 proinsulin, 364–365 prokaryote, 559 prolactin, 341, 346 prol ...